HU-243
 | |
| Identifiers | |
|---|---|
| |
| CAS Number |
140835-18-3  |
| PubChem (CID) | 3081854 |
| IUPHAR/BPS | 735 |
| Chemical and physical data | |
| Formula | C25H40O3 |
| Molar mass | 388.30 g/mol |
| 3D model (Jmol) | Interactive image |
| |
HU-243 (AM-4056) is a synthetic cannabinoid drug that is a single enantiomer of the hydrogenated derivative of the commonly used reference agonist HU-210. It is a potent agonist at both the CB1 and CB2 receptors, with a binding affinity of 0.041 nM at the CB1 receptor, making it marginally more potent than HU-210, which had an affinity of 0.061 nM in the same assay.[1]
See also
References
- ↑ Stern, E.; Lambert, D. M. (2007). "Medicinal Chemistry Endeavors around the Phytocannabinoids". Chemistry & Biodiversity. 4 (8): 1707–1728. doi:10.1002/cbdv.200790149. PMID 17712816.
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